 Product | | Comments |
| Bisindolylmaleimide Inhibitor Set | | A set of 6 separate vials. Each set contains 250 mg each of : - Bisindolylmaleimide I, HCl (Cat. No. 203291)
- Bisindolylmaleimide II (Cat. No. 203292)
- Bisindolylmaleimide III, HCl (Cat. No. 203294)
- Bisindolylmaleimide IV (Cat. No. 203297)
- Bisindolylmaleimide V (Cat. No. 203303)
- RIM-1 (Cat. No. 557325)
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| Calpain Inhibitor Set | | Provided as a 5 vial set. Each set contains: - 5 mg ALLN (Cat. No. 208719)
- 25 mg Calpain Inhibitor III (Cat. No. 208722)
- 5 mg of Calpeptin (Cat. No. 03-34-0051)
- 1 mg of EST (Cat. No. 330005)
- 5 mg of PD 150606 (Cat. No. 513022).
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| Caspase Inhibitor Set I | | The set of 3 separate vials. Each set contains 1 mg of: - Caspase-3 Inhibitor II, Z-DEVD-FMK (Cat. No. 264155)
- Caspase-1 Inhibitor I, Ac-YVAD-CHO (Cat. No. 400010)
- Caspase Inhibitor I, Z-VAD-FMK (Cat. No. 627610).
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| Caspase Inhibitor Set II | | The set of 8 separate vials. Each set contains 250 mg of: - Caspase-1 Inhibitor VI, Z-YVAD-FMK (Cat. No. 218746)
- Caspase-2 Inhibitor I, Z-VDVAD-FMK (Cat. No. 218744)
- Caspase-3 Inhibitor II, Z-DEVD-FMK (Cat. No. 264155)
- Caspase-5 Inhibitor I, ZWEHD- FMK (Cat. No. 218753)
- Caspase-6 Inhibitor I, Z-VEIDFMK (Cat. No. 218757)
- Caspase-8 Inhibitor II, Z-IETD-FMK (Cat. No. 218759)
- Caspase-9 Inhibitor I, Z-LEHD-FMK (Cat. No. 218761)
- Caspase Inhibitor III, Boc-D-FMK (Cat. No. 218745).
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| Caspase Inhibitor Set III | | A set of 8 separate vials. Each set contains a ready-to-use DMSO solution of irreversible inhibitors of various members of the caspase-family proteases. Contains 25 ml (2 mM) each of: - Caspase-1 Inhibitor VI, Z-YVAD-FMK (Cat. No. 218746)
- Caspase-2 Inhibitor I, Z-VDVAD-FMK (Cat. No. 218744)
- Caspase-3 Inhibitor II, Z-DEVD-FMK (Cat. No. 264155)
- Caspase-5 Inhibitor I, Z-WEHD-FMK (Cat. No. 218753)
- Caspase-6 Inhibitor I, Z-VEID-FMK (Cat. No. 218757)
- Caspase-8 Inhibitor II, Z-IETD-FMK (Cat. No. 218759)
- Caspase-9 Inhibitor I, Z-LEHD-FMK (Cat. No. 218761)
- Caspase Inhibitor I, Z-VAD-FMK (Cat. No. 627610).
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| Caspase Inhibitor Set IV | | A set of 6 separate vials. Each set contains a ready-to-use solution of reagents for caspase inhibition studies and an apoptosis inducer. Contains 25 ml of a 10 mM solution in DMSO of: - Caspase-3 Inhibitor II, Z-DEVD-FMK (Cat. No. 264155)
- Caspase-8 Inhibitor II, Z-IETD-FMK (Cat. No. 218759)
- Caspase-9 Inhibitor I, Z-LEHD-FMK (Cat. No 218761)
- General caspase inhibitor, Z-VAD-FMK (Cat. No. 627610)
- The negative control Z-FA-FMK (Cat. No. 342000)
- An aqueous solution (100 ml, 10.5 mM) of an apoptosis inducer, Doxorubicin, Hydrochloride (Cat. No. 324380).
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| Cyclin-Dependent Protein Kinase Inhibitor Set | | Provided as a 3 vial set. Each set contains: - 5 mg of Olomoucine (Cat. No. 495620)
- 1 mg of Iso-Olomoucine (Cat. No. 495622)
- 1 mg of Roscovitine (Cat. No. 557360)
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| Cyclooxygenase Inhibitor Set | | Provided as a 4 vial set. Each set contains: - 100 mg of Meloxicam (Cat. No. 444800)
- 5 mg of NS-398 (Cat. No. 349254)
- 5 mg of SC-560 (Cat. No. 565610)
- 5 mg of Sulindac Sulfide (Cat. No. 574102).
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| MAP Kinase Cascade Inhibitor Set | | A set of 5 vials. Each set contains: - 1 mg of FPT Inhibitor III (Cat. No. 344154)
- 1 mg of ZM 336372 (Cat. No. 692000)
- 5 mg of PD 98059 (Cat. No. 513000)
- 1 mg of SB 203580 (Cat. No. 559389)
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| MAP Kinase Inhibitor Set I | | A set of 4 vials. Each set contains: - 5 mg of the MEK inhibitor PD 98059 (Cat. No. 513000)
- 1 mg of the MAP kinase inhibitors SB 202190 (Cat. No. 559388)
- 1 mg of SB 203580 (Cat. No. 559389)
- 1 mg of the negative control, SB 202474 (Cat. No. 559387)
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| MAP Kinase Inhibitor Set II | | A set of 4 vials. Each set contains: - 5 mg of PD 98059 (Cat. No. 513000)
- 1 mg of SB 203580 (Cat. No. 559389)
- 1 mg of U0126 (Cat. No. 662005)
- 1 mg of the negative control, SB 202474 (Cat. No. 559387)
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| MEK Inhibitor Set | | A set of 3 vials. Each set contains: - 5 mg of PD 98059 (Cat. No. 513000)
- 1 mg of U0126 (Cat. No. 662005)
- 1 mg of the negative control U0124 (Cat. No. 662006)
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| MMP Inhibitor Set I | | Provided as a 5 vial set. Each set contains:
- 5 mg of MMP-2/MMP-9 Inhibitor I (Cat. No. 444241)
- 5 mg of MMP-3 Inhibitor II (Cat. No. 444225)
- 1 mg of GM 6001(Cat. No. 364205)
- 1 mg of GM 6001, Negative Control (Cat. No. 364210)
- 1 mg of MMP-8 Inhibitor I (Cat. No. 444237)
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| Nitric Oxide Synthase, Inducible, Inhibitor Set | | Provided as a 5 vial set. Each set contains: - 5 mg of 1400W (Cat. No. 100050)
- 10 mg of 1-Amino-2-hydroxyguanidine, p-Toluenesulfonate (Cat. No. 155200)
- 100 mg of S-Methylisothiourea Sulfate (Cat. No. 466220)
- 10 mg of L-NIL, Dihydrochloride (Cat. No. 482100)
- 50 mg of 1,3-PBITU, Dihydrobromide (Cat. No. 512774).
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| NOS Inhibitor Set | | Provided as a 6 vial set. Each set contains
- 20 mg of L-N5-(1-Iminoethyl)ornithine, HCl (Cat. No. 400600)
- 10 mg of S-Methyl-L-thiocitrulline, HCl (Cat. No. 472804)
- 25 mg of NG-Monomethyl-L-arginine, Monoacetate Salt (Cat. No. 475886)
- 100 mg of NG-Nitro-L-arginine Methyl Ester, HCl (Cat. No. 483125)
- 100 mg of NG-Nitro-D-arginine Methyl Ester, HCl, 100 mg of 7-Nitroindazole (Cat. No. 483400)
- 10 mg of L-Thiocitrulline, HCl (Cat. No. 589411)
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| PARP Inhibitor Set | | Provided as a 5 vial set. Each set contains - 100 mg of 3-Aminobenzamide (Cat. No. 165350)
- 5 mg of 5-Iodo-6-amino- 1,2-benzopyrone (Cat. No. 407850)
- 5 mg of 1,5-Isoquinolinediol (Cat. No. 419800)
- 5 mg of NU 1025 (Cat. No. 493800)
- 1 mg of DPQ (Cat. No. 300270)
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| Phosphodiesterase Inhibitor Set I | | Provided as a set of 4 vials. Each set contains: - 10 mg of 8-Methoxymethyl-3- isobutyl-1-methylxanthine (Cat. No. 454202), a Ca2+/CaM-dependent PDE (PDE I) inhibitor
- 1 mg of 4-{[3,4 -(Methylenedioxy)benzyl]amino}-6-methoxyquinazoline (Cat. No. 475250), a cGMP-specific PDE (PDE V) inhibitor
- 5 mg of Rolipram (Cat. No. 557330), a cAMP-specific PDE (PDE IV) inhibitor
- 10 mg of Trequinsin, Hydrochloride (Cat. No. 382425), a cGMP-inhibited PDE (PDE III) inhibitor.
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| Phosphotyrosine Phosphatase Inhibitor Set (Vanadium) | | Provided as a set of 3 vials. Each set contains: - 5 g of Sodium Orthovanadate (Cat. No. 567540)
- 10 mg of bpV(phen) (Cat. No. 203695)
- 10 mg of mpV(pic) (Cat. No. 475950)
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| Proteasome Inhibitor Set I | | A set of three vials. Each set contains: - 1 mg of Proteasome Inhibitor I (Cat. No. 539160)
- 200 mg of Lactacystin (Cat. No. 426100)
- 1 mg of MG-132 (Cat. No. 474790).
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| Proteasome Inhibitor Set II | | A set of three vials. Each set contains: - 5 mg of ALLN (Cat. No. 208719)
- 100 mg of Epoxomicin (Cat. No. 324800)
- 100 mg of clasto-Lactacystin b-Lactone (Cat. No. 426102).
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| Protein Kinase C Inhibitor Set | | A set of 6 vials. Each set contains: - 250 mg of Bisindolylmaleimide I (Cat. No. 203290)
- 50 mg of Calphostin C, Cladosporium cladosporioides (Cat. No. 208725)
- 5 mg of Chelerythrine Chloride (Cat. No. 220285)
- 500 mg of Gö 6976 (Cat. No. 365250)
- 500 mg of Myristoylated Protein Kinase C Inhibitor 20-28, Cell-Permeable (Cat. No. 476480)
- 500 mg of Ro-32-0432 (Cat. No. 557525)
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| Protein Kinase Inhibitor Set | | A set of 6 vials. Each set contains: - 500 mg of Ro-31-8220 (Cat. No. 557520)
- 20 mg of Genistein (Cat. No. 345834)
- 1 mg of KN-93, Water-Soluble (Cat. No. 422711)
- 50 mg of KT5720 (Cat. No. 420320)
- 100 mg of Staurosporine, Streptomyces sp. (Cat. No. 569397)
- 1 mg of U0126 (Cat. No. 662005)
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| Serine/Threonine Kinase Inhibitor Set | | A set of 6 vials. Each set contains: - 250 mg of PKC inhibitor, Bisindolylmaleimide I (Cat. No. 203290)
- 1 mg of PKA inhibitor, H-89, Dihydrochloride (Cat. No. 371963)
- 1 mg of PKG inhibitor, Protein Kinase G Inhibitor (Cat. No. 370654)
- 1 mg of MLCK inhibitor, ML-7 (Cat. No. 475880)
- 1 mg of CaM kinase II inhibitor, KN-93 (Cat. No. 422708)
- 100 mg of the broad range inhibitor, Staurosporine (Cat. No. 569397) Not available for sale in Japan.
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| Src Family Protein Tyrosine Kinase Inhibitor Set | | A set of 4 vials. Each set contains: - 20 mg of Genistein (Cat. No. 345834)
- 100 mg of Herbimycin A, Streptomyces sp. (Cat. No. 375670)
- 1 mg of PP2 (Cat. No. 529573)
- 1 mg of PP3 (Cat. No. 529574)
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| Tyrosine Kinase Inhibitor Set II | | A set of 4 vials. Each set contains: - 20 mg of Genistein (Cat. No. 345834)
- 1 mg of PP2 (Cat. No. 529573)
- 5 mg of AG 490 (Cat. No. 658401)
- 5 mg of AG 1296 (Cat. No. 658551)
- 5 mg of AG 1478 (Cat. No. 658552)
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