2-[1-(3-Aminopropyl)-1H-indol-3-yl]-3-(1H-indol-3-yl)maleimide, HCl Red solid. A potent, cell permeable, and selective inhibitor of protein kinase C (IC50 = 26 nM). May inhibit protein kinase A at much higher concentrations (IC50 = 500 nM). Purity: ≥95% by HPLC. Ref.: Fabre, S., and Prudhomme, M. 1993. Bioorg. Med. Chem. 1, 193. Davis, P.D., et al. 1992. J. Med. Chem. 35, 177. Toullec, D., et al. 1991. J. Biol. Chem. 266, 15771.
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