(N-Cyclopropyl-N-piperidin-4-yl)-4-chlorobenzenesulfonamide White solid. PROTECT FROM LIGHT. PACKAGED UNDER INERT GAS. A cell-permeable sulfonamide compound that reversibly interacts with the benzothiazepine-binding site and acts as a cardiac tissue selective L-type voltage gated Ca2+-channel activity inhibitor. Shown to display negative chronotropic activity with minimal vasorelaxation. Purity: ≥95% by HPLC. Ref.: Carosati, E., et al. 2006. J. Med. Chem. 49, 5206. |