a-4-Dibromoacetophenone
Tau Protein Kinase I Inhibitor
TPK I Inhibitor White solid. PROTECT FROM LIGHT. PROTECT FROM MOISTURE. PACKAGED UNDER INERT GAS. A phenyl a-bromomethyl ketone compound that acts as a cell-permeable, and non-ATP competitive inhibitor of GSK-3b (IC50 = 0.5 µM). This reactive alkylating agent is selective towards GSK-3b and does not affect PKA activity even at concentrations as high as 100 µM. Purity: ≥95% by HPLC. RTECS AM6950000, CAS 99-73-0. Ref.: Conde, S., et al. 2003. J. Med. Chem. 46, 4631. | 
