Off-white solid. PROTECT FROM LIGHT. PACKAGED UNDER INERT GAS. A cell-permeable, potent, selective, and reversible MMP-9 Inhibitor (IC50 = 5 nM). Inhibits MMP-1 (IC50 = 1.05 µM) and MMP-13 (IC50 = 113 nM) only at much higher concentrations. Purity: ≥95% by HPLC. Ref.: Levin, J.I., et al. 2001. Bioorg. Med. Chem. Lett. 11, 2189. |