H-Trp-Glu-OH White solid. PROTECT FROM LIGHT. PACKAGED UNDER INERT GAS. A cell-permeable dipeptide that acts as a selective and reversible PPARg antagonist (KD ~ 8 µM). Shown to inhibit the agonist activity of Rosiglitazone (100 nM) in a dose-dependent manner (IC50 = 31.9 µM) in transfected COS-7 cells. Purity: ≥97% by elemental analysis. CAS 36099-95-3. Ref.: Ye, F., et al. 2006. Chembiochem 7, 74. |